中文名称:HIF1AN抗原(重组蛋白)英文名称:HIF1AN Antigen (Recombinant Protein)别 名:FIH1储 存:冷冻(-20℃)相关类别:抗原概述Full length fusion protein技术规格
Full name:
hypoxia inducible factor 1, alpha subunit inhibitor
Synonyms:
FIH1
Swissprot:
Q9NWT6
Gene Accession:
BC007719
Purity:
>85%, as determined by Coomassie blue stained SDS-PAGE
Expression system:
Escherichia coli
Tags:
His tag C-Terminus, GST tag N-Terminus
Background:
Hydroxylates HIF-1 alpha at 'Asp-803' in the C-terminal transactivation domain (CAD). Functions as an oxygen sensor and, under normoxic conditions, the hydroxylation prevents interaction of HIF-1 with transcriptional coactivators including Cbp/p300-interacting transactivator. Involved in transcriptional repression through interaction with HIF1A, VHL and histone deacetylases. Hydroxylates specific Asn residues within ankyrin repeat domains (ARD) of NFKB1, NFKBIA, NOTCH1, ASB4, PPP1R12A and several other ARD-containing proteins. Also hydroxylates Asp and His residues within ARDs of ANK1 and TNKS2, respectively.
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